|T000068, COQ8A Tracer (PBI 6948)
Compound Image

T000068

COQ8A Tracer (PBI 6948)


  • Description

    Formula:

    C49H52BCl2F2N9O8

    avg. MolWt:

    1014.72 u

    PAINS elements:

    none detected

    SMILES:

    display
  • Properties

    Store at:

    -80 °C

    Absorption:

    450 nm

    Emission:

    590 nm

    clogP:

    6.52
  • References

    Contributing Lab:

    Promega Corp., Madison

  • Experimental

    : 2.21

    Z’: 0.86

    : yes

    Tracer titration

    KDapp:

    1792 nM
    ...
    raw data
    Tracer displacement
    i

    Compound used for displacement:

    PD173955

    EC50:

    642 nM
    raw data

    Comment: NLuc-COQ8A