|T000065, K14 Tracer
Compound Image

T000065

K14 Tracer


  • Properties

    Store at:

    -80 °C

    Absorption:

    450 nm

    Emission:

    590 nm
  • References

    Contributing Lab:

    Promega Corp., Madison and Knapp Lab, Knapp Lab, University of Frankfurt

  • Experimental

    : 9.1

    Z’: 0.95

    : yes

    Tracer titration

    KDapp:

    2457 nM
    ...
    raw data
    Tracer displacement
    i

    Compound used for displacement:

    Vactosertib

    EC50:

    267 nM
    raw data

    Comment: ACVR1B/ALK4-NLuc

    Reference: PMID

    : 8.4

    Z’: 0.96

    : yes

    Tracer titration

    KDapp:

    1523 nM
    ...
    raw data
    Tracer displacement
    i

    Compound used for displacement:

    Vactosertib

    EC50:

    367 nM
    raw data

    Comment: TGFβR1/ALK5-NLuc

    Reference: PMID