|T000006, WDR5 Tracer
Compound Image

T000006

WDR5 Tracer

  • Description

    Formula:

    C51H57BF5N9O7

    avg. MolWt:

    1013.87 u

    PAINS elements:

    none detected

    SMILES:

    display
  • Properties

    Store at:

    -80 °C

    Absorption:

    450 nm

    Emission:

    590 nm

    clogP:

    6.15
  • References

    Synthesis:

    Publication

    Contributing Lab:

    Knapp Lab, University of Frankfurt

  • Experimental

    : 2.2

    Z’: 0.6

    : yes

    Tracer titration

    KDapp:

    2812 nM
    ...
    raw data
    Tracer displacement
    i

    Compound used for displacement:

    OICR-9429

    EC50:

    339 nM
    raw data

    Reference: PMID