|T000032, PBI 9191
Compound Image

T000032

PBI 9191

  • Description

    Formula:

    C42H49BClF2N13O2

    avg. MolWt:

    852.2 u

    PAINS elements:

    none detected

    SMILES:

    display
  • Properties

    Store at:

    -80 °C

    Absorption:

    450 nm

    Emission:

    590 nm

    clogP:

    6.37
  • References

    Synthesis:

    Publication

    Contributing Lab:

    Promega Corp., Madison

  • Experimental

    : 2.9

    Z’: 0.95

    : yes

    Tracer titration

    KDapp:

    225 nM
    ...
    raw data
    Tracer displacement
    i

    Compound used for displacement:

    Danusertib

    EC50:

    146 nM
    raw data

    Comment: AURKA-NLuc

    Reference: PMID